SCHEMBL30007416

SCHEMBL30007416

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)c(Cl)c(-c3ccc(F)cc3)n2)C2CC2)cc2cc(C)cnc12

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.34
CFTR P13569 3/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ROCK2 O75116 3/20 0.32
ROCK1 Q13464 3/20 0.32
GABRA5 P31644 2/20 0.32
RIPK1 Q13546 3/20 0.32
MCHR1 Q99705 2/20 0.31
HTR2C P28335 1/20 0.31
MAPT P10636 1/20 0.31
GRIN2B Q13224 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25687220 1.00 CNR1 (0.34) CNR1CFTRKDM4EALDH1A1HTT
SCHEMBL25279914 1.00 CNR1 (0.34) CNR1CFTRKDM4EALDH1A1HTT
SCHEMBL25687225 0.94 CFTR (0.35) CNR1CFTRALDH1A1NPSR1RXFP1
SCHEMBL30006884 0.93 CNR1 (0.34) CNR1CFTRGABRA5MCHR1HTR2C
SCHEMBL25687285 0.93 CNR1 (0.34) CNR1CFTRGABRA5MCHR1HTR2C
SCHEMBL28909199 0.92 CFTR (0.36) CNR1CFTRROCK2ROCK1RIPK1
SCHEMBL25687507 0.92 CFTR (0.36) CNR1CFTRROCK2ROCK1RIPK1
SCHEMBL30007164 0.91 P2RX7 (0.33) CNR1CFTRALDH1A1ROCK2ROCK1
SCHEMBL25687297 0.91 P2RX7 (0.33) CNR1CFTRALDH1A1ROCK2ROCK1
SCHEMBL25233253 0.91 CNR1 (0.39) CNR1KDM4EALDH1A1HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed