SCHEMBL30007164

SCHEMBL30007164

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)c(Cl)c(-c3ccc(F)cc3)n2)C2CC2)cc2cc(C(F)F)cnc12

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.33
CNR1 P21554 1/20 0.33
CFTR P13569 3/20 0.33
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
RIPK1 Q13546 5/20 0.32
KCNH2 Q12809 2/20 0.31
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ROCK2 O75116 2/20 0.31
ROCK1 Q13464 2/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25687297 1.00 P2RX7 (0.33) P2RX7CNR1CFTRLMNATP53
SCHEMBL30007232 0.94 CFTR (0.34) P2RX7CNR1CFTRLMNATP53
SCHEMBL25687300 0.94 CFTR (0.34) P2RX7CNR1CFTRLMNATP53
SCHEMBL25279914 0.91 CNR1 (0.34) CNR1CFTRRIPK1ALDH1A1ROCK2
SCHEMBL30007416 0.91 CNR1 (0.34) CNR1CFTRRIPK1ALDH1A1ROCK2
SCHEMBL25687220 0.91 CNR1 (0.34) CNR1CFTRRIPK1ALDH1A1ROCK2
SCHEMBL28909199 0.90 CFTR (0.36) P2RX7CNR1CFTRRIPK1ROCK2
SCHEMBL25687507 0.90 CFTR (0.36) P2RX7CNR1CFTRRIPK1ROCK2
SCHEMBL30007273 0.89 CFTR (0.33) P2RX7CNR1CFTRLMNATP53
SCHEMBL25687403 0.89 CFTR (0.33) P2RX7CNR1CFTRLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed