SCHEMBL30007553

SCHEMBL30007553

O=c1[nH]c(C(F)F)nc2cnc(Br)cc12

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
HCAR2 Q8TDS4 9/20 0.37
ROCK2 O75116 6/20 0.32
ROCK1 Q13464 2/20 0.32
GPR39 O43194 1/20 0.31
KDM5A P29375 1/20 0.31
KDM4C Q9H3R0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101302 0.77 GAA (0.51) ALDH1A1POLBROCK2
SCHEMBL24625406 0.76 KDM4E (0.53) ALDH1A1POLB
SCHEMBL30754559 0.76 KDM5A (0.56) ALDH1A1POLBHCAR2KDM5AKDM4C
SCHEMBL11782173 0.73 HCAR2 (0.43) ALDH1A1POLBHCAR2
SCHEMBL25098508 0.73 HCAR2 (0.37) ALDH1A1POLBHCAR2ROCK1
SCHEMBL24791096 0.71 GRIN2D (0.44) ALDH1A1POLB
SCHEMBL24792669 0.70 KDM4E (0.52) ALDH1A1POLB
SCHEMBL30170779 0.70 KDM4E (0.52) ALDH1A1POLB
SCHEMBL22101792 0.68 PIM1 (0.38) HCAR2
SCHEMBL24792663 0.66 GUSB (0.43) ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119894893-A Sulfone substituted pyrido [3,4-D ] pyrimidine derivatives for the treatment of cancer 拜耳公司 2025-04-25 CN disclosed
EP-4322962-A1 PHOSPHORUS DERIVATIVES AS NOVEL SOS1 INHIBITORS Bayer Aktiengesellschaft (DE) 2024-02-21 EP disclosed
CN-117500507-A Phosphorus derivatives as novel SOS1 inhibitors 拜耳公司 2024-02-02 CN disclosed
WO-2022219035-A1 PHOSPHORUS DERIVATIVES AS NOVEL SOS1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2022-10-20 WO disclosed