SCHEMBL30007857

SCHEMBL30007857

CC(C)c1cc(C(=O)NN)ccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
MPO P05164 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP1A2 P05177 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2A6 P11509 1/20 0.50
CYP2C19 P33261 1/20 0.50
ALDH1A1 P00352 1/20 0.42
RAF1 P04049 7/20 0.41
BRAF P15056 7/20 0.41
PROKR1 Q8TCW9 1/20 0.41
FDPS P14324 1/20 0.40
MAPT P10636 1/20 0.40
P2RX7 Q99572 2/20 0.39
KDM5A P29375 1/20 0.39
BLM P54132 1/20 0.39
GFER P55789 1/20 0.39
PMP22 Q01453 1/20 0.39
HIF1A Q16665 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4000772 1.00 KDM4E (0.50) KDM4EMPOCYP3A4CYP1A2ADORA3
SCHEMBL14566838 0.85 PLK1 (0.46) RAF1BRAFPROKR1FDPSKDM5A
SCHEMBL25820303 0.83 FDPS (0.57) CYP3A4ALDH1A1RAF1BRAFPROKR1
SCHEMBL23015656 0.81 HPGD (0.48) KDM4EADORA3ALDH1A1MAPTKDM5A
SCHEMBL21212289 0.81 GAA (0.46) RAF1BRAFKMT2A
SCHEMBL30418990 0.81 KDM5C (0.44) CYP3A4CYP1A2PROKR1KDM5A
SCHEMBL6047032 0.81 KDM5C (0.44) CYP3A4CYP1A2PROKR1KDM5A
SCHEMBL1759894 0.79 KDM4C (0.55) KDM4EALDH1A1PROKR1MAPTKDM5A
SCHEMBL25905366 0.79 PROKR1 (0.44) KDM4ECYP3A4CYP1A2CYP2A6ALDH1A1
SCHEMBL8953772 0.78 KDM4E (0.57) KDM4ECYP3A4CYP1A2ALDH1A1PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110234638-B Heteroaryl phenoxy benzamide KAPPA opioid ligands 辉瑞大药厂 2022-10-21 CN disclosed