SCHEMBL3000928

SCHEMBL3000928

COc1ncc(B2OC(C)(C)C(C)(C)O2)cc1/C=C/c1ccc(N2CCN(C(=O)O)CC2)cc1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.38
CYP17A1 P05093 8/20 0.38
CYP21A2 P08686 8/20 0.38
CYP11B1 P15538 8/20 0.38
CYP3A4 P08684 1/20 0.36
CYP19A1 P11511 1/20 0.36
MAPT P10636 2/20 0.36
P4HB P07237 1/20 0.35
ACHE P22303 5/20 0.35
ALPL P05186 1/20 0.35
ALK Q9UM73 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3000938 1.00 MAOB (0.38) MAOBCYP17A1CYP21A2CYP11B1CYP3A4
SCHEMBL1136795 0.89 ABCB1 (0.46) MAPTALK
SCHEMBL1136797 0.89 ABCB1 (0.46) MAPTALK
SCHEMBL1136842 0.82 ALPL (0.32) MAOBCYP17A1CYP21A2CYP11B1P4HB
SCHEMBL1136850 0.82 ALPL (0.32) MAOBCYP17A1CYP21A2CYP11B1P4HB
SCHEMBL1136702 0.81 CYP17A1 (0.41) CYP17A1CYP21A2CYP11B1CYP3A4CYP19A1
SCHEMBL1136704 0.81 CYP17A1 (0.41) CYP17A1CYP21A2CYP11B1CYP3A4CYP19A1
SCHEMBL578443 0.74 LIPG (0.44) P4HB
SCHEMBL1136706 0.73 MAPT (0.44) MAOBMAPTACHEALK
SCHEMBL1136707 0.73 MAPT (0.44) MAOBMAPTACHEALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7786120-B2 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-08-31 US disclosed
US-20070185125-A1 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED 2007-08-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185125-A1 Pyridones useful as inhibitors of kinases MAP3K20, MAP3K6, MAP3K5 MAOB 912/4885CYP17A1 3080/4885CYP21A2 3083/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.