SCHEMBL30009609

SCHEMBL30009609

C#Cc1ccc2c3c([nH]c2c1)C(C)(C)c1cc(N2CCC(N4CCOCC4)CC2)c(Cl)cc1C3

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 20/20 0.61
KDR P35968 4/20 0.52
KIT P10721 3/20 0.52
GAK O14976 1/20 0.51
ACOX3 O15254 1/20 0.51
NR1I2 O75469 1/20 0.51
ABCB11 O95342 1/20 0.51
EGFR P00533 1/20 0.51
ESR1 P03372 1/20 0.51
PGR P06401 1/20 0.51
RET P07949 1/20 0.51
ROS1 P08922 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
PHKG2 P15735 1/20 0.51
FER P16591 1/20 0.51
EPHA1 P21709 1/20 0.51
DRD1 P21728 1/20 0.51
SLC6A2 P23975 1/20 0.51
PDE4A P27815 1/20 0.51
SLC6A4 P31645 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30009076 0.91 ALK (0.50) ALKKDRKIT
SCHEMBL30010172 0.88 ALK (0.56) ALKKDRKITGAKACOX3
SCHEMBL30009674 0.84 ALK (0.46) ALKKDRKITSRPK2SRPK1
SCHEMBL28960837 0.84 ALK (0.85) ALKKDRKITGAKACOX3
SCHEMBL20004242 0.82 ALK (0.62) ALKKDRKITGAKACOX3
SCHEMBL20634798 0.81 ALK (0.74) ALKKDRKITGAKACOX3
SCHEMBL28960826 0.78 ALK (0.57) ALKKDRKITGAKACOX3
SCHEMBL30009083 0.78 ALK (0.44) ALKKDRKIT
SCHEMBL27087552 0.77 ALK (0.72) ALKKDRKITGAKACOX3
SCHEMBL27087532 0.77 ALK (0.77) ALKKDRKITGAKACOX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237813-A1 COMPOUND HAVING ALK INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 盛世泰科生物医药技术(苏州)有限公司 2022-11-17 WO disclosed