SCHEMBL30016319

SCHEMBL30016319

CNc1ccnc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 1/20 0.51
SMARCA4 P51532 1/20 0.51
LOXL2 Q9Y4K0 2/20 0.47
LOX P28300 1/20 0.46
TAS2R14 Q9NYV8 1/20 0.43
IDH2 P48735 4/20 0.42
IDH1 O75874 3/20 0.42
NOTUM Q6P988 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9234478 1.00 SMARCA2 (0.51) SMARCA2SMARCA4LOXL2LOXTAS2R14
SCHEMBL22601563 0.82 PRKCI (0.49) SMARCA2SMARCA4IDH2IDH1HDAC4
SCHEMBL27893424 0.80 KIF11 (0.53) LOXL2NOTUM
SCHEMBL2479367 0.80 LOXL2 (0.52) SMARCA2SMARCA4LOXL2LOXTAS2R14
SCHEMBL30505955 0.80 LOXL2 (0.52) SMARCA2SMARCA4LOXL2LOXTAS2R14
SCHEMBL23639222 0.80 SMARCA2 (0.51) SMARCA2SMARCA4LOXL2LOXTAS2R14
SCHEMBL25124381 0.79 SMARCA2 (0.48) SMARCA2SMARCA4LOXL2LOXTAS2R14
Hydrochloric Acid SCHEMBL16633226 0.78 LOXL2 (0.53) SMARCA2SMARCA4LOXL2LOXTAS2R14
Hydrochloric Acid SCHEMBL31696645 0.78 LOXL2 (0.53) SMARCA2SMARCA4LOXL2LOXTAS2R14
SCHEMBL24258152 0.77 SMARCA2 (0.64) SMARCA2SMARCA4HDAC4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113264945-B Spiro derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed