SCHEMBL300458

SCHEMBL300458

CCN(CC)c1ccc2c(c1)Oc1cc3c(cc1C2(O)c1ccccc1C=O)C1(OC(=O)c2ccccc21)c1ccc(N(CC)CC)cc1O3

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.48
FTO Q9C0B1 5/20 0.47
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
MAPT P10636 4/20 0.47
HTT P42858 2/20 0.47
HPGD P15428 2/20 0.47
RECQL P46063 2/20 0.47
BLM P54132 2/20 0.47
PRMT1 Q99873 2/20 0.47
ACE2 Q9BYF1 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
CYP2C19 P33261 1/20 0.47
SMAD3 P84022 1/20 0.47
ALDH1A1 P00352 4/20 0.45
LMNA P02545 2/20 0.45
USP2 O75604 2/20 0.45
CA12 O43570 4/20 0.41
CA1 P00915 4/20 0.41
CA2 P00918 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300176 0.91 CYP3A4 (0.45) CYP3A4FTOMEN1KMT2AMAPT
SCHEMBL275739 0.87 CYP3A4 (0.60) CYP3A4FTOMEN1KMT2AMAPT
SCHEMBL13069672 0.86 ALDH1A1 (0.46) MEN1KMT2AMAPTHTTHPGD
SCHEMBL21440424 0.84 CYP3A4 (0.61) CYP3A4FTOMEN1KMT2AMAPT
SCHEMBL31150744 0.84 CYP3A4 (0.64) CYP3A4FTOMEN1KMT2AMAPT
SCHEMBL29369814 0.84 CYP3A4 (0.64) CYP3A4FTOMEN1KMT2AMAPT
SCHEMBL52075 0.84 CYP3A4 (0.64) CYP3A4FTOMEN1KMT2AMAPT
SCHEMBL9104715 0.82 CYP3A4 (0.59) CYP3A4FTOMEN1KMT2AMAPT
SCHEMBL10347973 0.82 CYP3A4 (0.61) CYP3A4FTOMEN1KMT2AMAPT
SCHEMBL11882058 0.82 CYP3A4 (0.52) CYP3A4FTOMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134017-B1 Compound and use thereof RIKEN (JP) 2012-03-13 US disclosed