SCHEMBL30068660

SCHEMBL30068660

Brc1cc2c(c(Cc3ccccc3)c1)COCC2

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTRC Q99895 1/20 0.35
CCR5 P51681 1/20 0.34
BCL2 P10415 1/20 0.34
BCL2L1 Q07817 1/20 0.34
ALOX5 P09917 1/20 0.34
LMNA P02545 1/20 0.33
BRD4 O60885 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
SLC5A2 P31639 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
CALM1 P0DP23 1/20 0.31
HTR2B P41595 2/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25260735 0.77 ALDH1A1 (0.30)
SCHEMBL30068862 0.77 ALDH1A1 (0.30)
SCHEMBL30068919 0.77 MAPK1 (0.35) LMNA
SCHEMBL25260744 0.74 CSNK2A1 (0.31)
SCHEMBL25260922 0.74 KDM4E (0.42) CCR5LMNA
SCHEMBL25302681 0.72 MAPT (0.46)
SCHEMBL25296632 0.71 MAPT (0.44) CCR5LMNA
SCHEMBL25254901 0.71 TSHR (0.45) CCR5
SCHEMBL25256658 0.71 CYP2A13 (0.44) CCR5
SCHEMBL25296297 0.71 WNT3A (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022184152-A1 FUSED RING SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2022-09-09 WO disclosed