SCHEMBL300705

SCHEMBL300705

O=C=Nc1ccccc1C(c1ccccc1)c1ccccc1N=C=O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 3/20 0.33
ALDH1A1 P00352 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
TRPA1 O75762 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
CFTR P13569 1/20 0.31
GOPC Q9HD26 1/20 0.31
CYP2D6 P10635 1/20 0.30
MIF P14174 1/20 0.30
SRC P12931 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365140 0.88 CYP3A4 (0.50) CYP3A4ALDH1A1TDP1TRPA1MIF
SCHEMBL11468798 0.87 CYP3A4 (0.40) CYP3A4ALDH1A1TDP1GAAKMT2A
SCHEMBL374655 0.84 CYP3A4 (0.40) CYP3A4ALDH1A1TDP1GAAKMT2A
SCHEMBL15738978 0.82 CYP3A4 (0.45) CYP3A4ALDH1A1TDP1TRPA1HPGD
SCHEMBL28036817 0.82 CYP3A4 (0.43) CYP3A4ALDH1A1TDP1GAAKMT2A
SCHEMBL30378062 0.80 CYP3A4 (0.40) CYP3A4MIF
SCHEMBL4651380 0.80 CYP3A4 (0.40) CYP3A4MIF
SCHEMBL4669249 0.80 CYP3A4 (0.41) CYP3A4ALDH1A1TDP1KMT2ATRPA1
SCHEMBL2836253 0.79 CYP3A4 (0.47) CYP3A4SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL532582 0.79 CYP3A4 (0.42) CYP3A4ALDH1A1TDP1TRPA1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010588-B1 Organosilicon polyurea polymers, elastomers manufactured therefrom and their use HENKEL AG & CO KGAA (DE) 2012-01-04 EP claimed
EP-0111259-B1 PROCESS FOR THE PREPARATION OF COMPOUNDS CONTAINING (METH)ACRYLIC-ACID ESTERS, (METH)ACRYLIC-ACID ESTERS AND ANAEROBICALLY CURABLE ADHESIVES AND PUTTY-LIKE MASSES Henkel Kommanditgesellschaft auf Aktien (DE) 1988-05-25 EP claimed
EP-0111259-A2 Process for the preparation of compounds containing (meth)acrylic-acid esters, (meth)acrylic-acid esters and anaerobically curable adhesives and putty-like masses Henkel Kommanditgesellschaft auf Aktien (DE) 1984-06-20 EP claimed
WO-2020225088-A1 METHOD FOR THE PURIFICATION OF ISOCYANATES COVESTRO INTELLECTUAL PROPERTY GMBH & CO. KG (DE) 2020-11-12 WO disclosed
EP-3736263-A1 METHOD FOR THE PURIFICATION OF ISOCYANATES Covestro Deutschland AG (DE) 2020-11-11 EP disclosed
EP-2794769-B9 PIGMENTED, FINE-STRUCTURED, TRIBOLOGICAL COMPOSITE MATERIAL LEIBNIZ INSTITUT FUER NEUE MAT GEMEINNUETZIGE GMBH (DE) 2019-03-20 EP disclosed
EP-2380061-B1 METHOD FOR PRODUCING OPTICAL ELEMENTS HAVING A GRADIENT STRUCTURE AND OPTICAL ELEMENT HAVING A GRADIENT STRUCTURE LEIBNIZ-INSTITUT FÜR NEUE MAT GEMEINNÜTZIGE GMBH (DE) 2017-12-06 EP disclosed
EP-2794769-B1 PIGMENTED, FINE-STRUCTURED, TRIBOLOGICAL COMPOSITE MATERIAL LEIBNIZ INST FÜR NEUE MATERIALIEN GEMEINNÜTZIGE GMBH (DE) 2016-09-14 EP disclosed
EP-2794769-A1 PIGMENTED, FINE-STRUCTURED, TRIBOLOGICAL COMPOSITE MATERIAL Leibniz-Institut für Neue Materialien gemeinnützige GmbH (DE) 2014-10-29 EP disclosed
WO-2013092835-A1 PIGMENTED, FINE-STRUCTURED, TRIBOLOGICAL COMPOSITE MATERIAL LEIBNIZ-INSTITUT FÜR NEUE MATERIALIEN GEMEINNÜTZIGE GMBH (DE) 2013-06-27 WO disclosed
EP-2245487-A1 OPTICAL ELEMENTS WITH GRADIENT STRUCTURE Leibniz-Institut für Neue Materialien gemeinnützige GmbH (DE) 2010-11-03 EP disclosed
US-4699866-A Preparation of electrostatographic encapsulated toner material improved in powder characteristics FUJI PHOTO FILM CO., LTD. (JP) 1987-10-13 US disclosed
US-4476211-A Preparation of electrostatographic toner material provided with surface electroconductivity FUJI PHOTO FILM CO., LTD. (JP) 1984-10-09 US disclosed
US-4468446-A Electrostatographic encapsulated toner material improved in powder characteristics FUJI PHOTO FILM CO., LTD. (JP) 1984-08-28 US disclosed
US-4465756-A Electrostatographic enscapsulated toner material improved in chargeability FUJI PHOTO FILM CO., LTD. (JP) 1984-08-14 US disclosed
US-4465755-A Pressure fixable electrostatographic toner material comprising encapsulated particles containing curing agent FUJI PHOTO FILM CO., LTD. 1984-08-14 US disclosed
EP-0111259-A2 Process for the preparation of compounds containing (meth)acrylic-acid esters, (meth)acrylic-acid esters and anaerobically curable adhesives and putty-like masses Henkel Kommanditgesellschaft auf Aktien (DE) 1984-06-20 EP disclosed
US-4455362-A Preparation of encapsulated electrostatographic toner material FUJI PHOTO FILM CO., LTD. (JP) 1984-06-19 US disclosed
US-4336308-A Magnetic recording media FUJI PHOTO FILM CO., LTD. (JP) 1982-06-22 US disclosed
US-4272585-A TO IMPROVE ADHESION, COATING WITH POLYURETHANE OR ALKYL POLYMETHACRYLATE IN POLAR APROTIC SOLVENT PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1981-06-09 US disclosed