SCHEMBL30085539

SCHEMBL30085539

Clc1ccc(-c2cc(N3CCN(CCN4CCOCC4)CC3)nc(-c3cccnc3)n2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.60
CYP2D6 P10635 4/20 0.60
CYP2C9 P11712 4/20 0.60
CYP2C19 P33261 4/20 0.60
PIK3CA P42336 4/20 0.59
PIK3CB P42338 2/20 0.58
PIK3CG P48736 2/20 0.58
CYP1A2 P05177 3/20 0.54
MAPT P10636 2/20 0.53
TSHR P16473 1/20 0.53
MAPK1 P28482 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HSD17B10 Q99714 1/20 0.53
ROS1 P08922 4/20 0.50
AIMP2 Q13155 1/20 0.49
MTOR P42345 1/20 0.48
PDE10A Q9Y233 1/20 0.48
SLC2A1 P11166 1/20 0.48
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28894649 1.00 CYP3A4 (0.60) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL30085536 0.92 PIK3CA (0.69) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL28895000 0.92 PIK3CA (0.69) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL30085495 0.90 CYP3A4 (0.48) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL28894723 0.90 CYP3A4 (0.48) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL28894647 0.89 PIM1 (0.49) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL30085814 0.89 PIM1 (0.49) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL30085626 0.86 TSHR (0.53) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL28895015 0.86 TSHR (0.53) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA
SCHEMBL28894784 0.86 P4HTM (0.49) CYP3A4CYP2D6CYP2C9CYP2C19PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN claimed
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN disclosed