SCHEMBL30100329

SCHEMBL30100329

NC(=O)c1ccc2nc(C(F)(F)F)cn2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 1/20 0.47
MCHR1 Q99705 9/20 0.46
CHEK1 O14757 1/20 0.45
AURKA O14965 1/20 0.45
DAPK3 O43293 1/20 0.45
JAK2 O60674 1/20 0.45
PRKD3 O94806 1/20 0.45
MAP4K4 O95819 1/20 0.45
PAK4 O96013 1/20 0.45
ABL1 P00519 1/20 0.45
NTRK1 P04629 1/20 0.45
FYN P06241 1/20 0.45
CSF1R P07333 1/20 0.45
RET P07949 1/20 0.45
MET P08581 1/20 0.45
PDGFRB P09619 1/20 0.45
PIM1 P11309 1/20 0.45
FGFR1 P11362 1/20 0.45
PDGFRA P16234 1/20 0.45
PRKACA P17612 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16739619 0.86 KDM4E (0.50) SCN5AMCHR1CCNB2CCNE2CDK1
SCHEMBL10311041 0.84 MCHR1 (0.52) MCHR1CHEK1AURKADAPK3JAK2
SCHEMBL38662516 0.79 MCHR1 (0.53) SCN5AMCHR1KDM4EALDH1A1NPC1
SCHEMBL30845741 0.77 EGLN1 (0.52) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL10053505 0.76 MCHR1 (0.48) MCHR1CHEK1AURKADAPK3JAK2
SCHEMBL18080888 0.75 SCN5A (0.53) SCN5AMCHR1TGFBR1KDM4EALDH1A1
SCHEMBL327269 0.74 PTGS1 (0.54) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL9570267 0.73 CHEK1 (0.46) MCHR1CHEK1AURKADAPK3JAK2
SCHEMBL9597339 0.73 MCHR1 (0.50) MCHR1CHEK1AURKADAPK3JAK2
SCHEMBL12056714 0.73 SCN5A (0.54) SCN5AMCHR1CDK5KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022255900-A1 CYSTEINYL LEUKOTRIENE RECEPTOR LIGANDS DIRECTED TOWARD THE TREATMENT OF INFLAMMATORY AND ONCOLOGICAL DISEASES федеральное государственное автономное образовательное учреждение высшего образования "Московский физико-технический институт (национальный исследовательский университет)" 2022-12-08 WO disclosed