SCHEMBL30103083

SCHEMBL30103083

COC(=O)c1cc(Cl)cc2cnn(Cc3ccc(-c4ccc(OC)c(F)c4)nc3)c12

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.41
CACNA1H O95180 7/20 0.41
PTGES O14684 1/20 0.38
MCHR1 Q99705 1/20 0.38
GRM2 Q14416 3/20 0.37
ROCK2 O75116 1/20 0.37
PKM P14618 1/20 0.37
PKLR P30613 1/20 0.37
P2RX3 P56373 2/20 0.36
MEN1 O00255 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
CNR1 P21554 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30103022 0.94 CACNA1H (0.41) BRD4CACNA1HGRM2ROCK2MEN1
SCHEMBL24785847 0.92 BRD4 (0.40) BRD4CACNA1HPTGESMCHR1GRM2
SCHEMBL30103081 0.92 BRD4 (0.40) BRD4CACNA1HPTGESMCHR1GRM2
SCHEMBL24785849 0.92 BRD4 (0.42) BRD4CACNA1HPTGESMCHR1GRM2
SCHEMBL30018129 0.90 BRD4 (0.41) BRD4CACNA1HMCHR1GRM2PKM
SCHEMBL24785366 0.90 BRD4 (0.41) BRD4CACNA1HMCHR1GRM2PKM
SCHEMBL24785813 0.88 GRIN2B (0.38) BRD4CACNA1HPTGESMCHR1GRM2
SCHEMBL30018152 0.88 GRIN2B (0.38) BRD4CACNA1HPTGESMCHR1GRM2
SCHEMBL30103066 0.86 CACNA1H (0.40) CACNA1HGRM2ROCK2MEN1KMT2A
SCHEMBL24785454 0.86 BRD4 (0.41) BRD4CACNA1HGRM2ROCK2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115448913-A Bicyclic compounds for the treatment of EP2, EP4 receptor mediated diseases 武汉人福创新药物研发中心有限公司 2022-12-09 CN disclosed