SCHEMBL3010334

SCHEMBL3010334

[c]1ccc(C2CCNCC2)cc1C1=CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 4/20 0.40
KIT P10721 1/20 0.40
QDPR P09417 1/20 0.38
HTR2C P28335 8/20 0.37
CYP2C9 P11712 1/20 0.36
SLC18A3 Q16572 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
PDE4B Q07343 1/20 0.30
TLR9 Q9NR96 1/20 0.30
TLR8 Q9NR97 1/20 0.30
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3005989 0.79 CSF1R (0.41) CSF1RQDPRHTR2CSLC18A3SIGMAR1
SCHEMBL18240960 0.77 CSF1R (0.45) CSF1RKITSLC18A3TLR9TLR8
SCHEMBL4380557 0.74 CSF1R (0.49) CSF1RKITTLR9TLR8TLR7
SCHEMBL4979196 0.74 CSF1R (0.49) CSF1R
SCHEMBL4057863 0.74 CSF1R (0.49) CSF1RKITHDAC1HDAC2TLR9
SCHEMBL2914743 0.74 CSF1R (0.49) CSF1RKITQDPRHTR2CCYP2C9
SCHEMBL3164538 0.73 CSF1R (0.48) CSF1RKITQDPRHTR2CCYP2C9
SCHEMBL18240980 0.72 CSF1R (0.41) CSF1RKITCYP2C9TLR9TLR8
SCHEMBL2914647 0.71 CSF1R (0.43) CSF1RKITCYP2C9HDAC1HDAC2
SCHEMBL2097686 0.70 QDPR (0.49) QDPRHTR2CSLC18A3SIGMAR1TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222298-A1 USE OF CFMS INHIBITOR FOR TREATING OR PREVENTING BONE CANCER AND THE BONE LOSS AND BONE PAIN ASSOCIATED WITH BONE CANCER Janssen Pharmaceutica N.V. (BE) 2010-09-01 EP disclosed
WO-2009058801-A1 USE OF CFMS INHIBITOR FOR TREATING OR PREVENTING BONE CANCER AND THE BONE LOSS AND BONE PAIN ASSOCIATED WITH BONE CANCER JANSSEN PHARMACEUTICA, N.V. (BE) 2009-05-07 WO disclosed
EP-1951234-A2 METHOD OF INHIBITING FLT3 KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-08-06 EP disclosed
WO-2007048088-A2 METHOD OF INHIBITING FLT3 KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2007-04-26 WO disclosed