SCHEMBL30107439

SCHEMBL30107439

CCc1ccncc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LPL P06858 6/20 0.40
LIPG Q9Y5X9 6/20 0.40
CYP2E1 P05181 4/20 0.40
CYP2C8 P10632 4/20 0.40
CYP2D6 P10635 4/20 0.40
CYP2A6 P11509 4/20 0.40
CYP2B6 P20813 4/20 0.40
CYP2C19 P33261 4/20 0.40
UCHL1 P09936 1/20 0.38
CYP2C9 P11712 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 1/20 0.36
F11 P03951 1/20 0.36
AOC1 P19801 4/20 0.35
AOC3 Q16853 4/20 0.35
PTGS1 P23219 2/20 0.32
PTGS2 P35354 1/20 0.32
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20517178 1.00 LPL (0.40) LPLLIPGCYP2E1CYP2C8CYP2D6
SCHEMBL24456240 0.87 LPL (0.37) LPLLIPGCYP2E1CYP2C8CYP2D6
SCHEMBL18356347 0.85 F11 (0.38) LPLLIPGUCHL1F11AOC1
SCHEMBL23295525 0.83 CYP11B1 (0.38) LPLLIPGUCHL1F11
SCHEMBL29542703 0.83 CYP11B1 (0.38) LPLLIPGUCHL1F11
SCHEMBL2352761 0.77 LPL (0.34) LPLLIPGCYP2E1CYP2C8CYP2D6
SCHEMBL29515710 0.77 LPL (0.34) LPLLIPGCYP2E1CYP2C8CYP2D6
SCHEMBL29572040 0.77 HTT (0.37) LPLLIPGCYP2E1CYP2C8CYP2D6
SCHEMBL4119052 0.77 HTT (0.37) LPLLIPGCYP2E1CYP2C8CYP2D6
SCHEMBL166233 0.76 GAA (0.34) LPLLIPGUCHL1F11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110678466-B Diazanaphthalenes as HPK1 inhibitors 豪夫迈·罗氏有限公司 2023-01-31 CN disclosed