SCHEMBL30107573

SCHEMBL30107573

Fc1cnc(Cl)nc1C#Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.43
FFAR1 O14842 1/20 0.42
APP P05067 1/20 0.40
ADORA2A P29274 1/20 0.39
GRM5 P41594 5/20 0.39
ADK P55263 1/20 0.38
CDK2 P24941 1/20 0.36
GRM4 Q14833 1/20 0.36
PTGES O14684 1/20 0.36
PIN1 Q13526 1/20 0.35
PLAU P00749 1/20 0.35
PLAT P00750 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24047399 1.00 MAPT (0.43) MAPTFFAR1APPADORA2AGRM5
SCHEMBL3442581 0.82 GRM5 (0.43) MAPTFFAR1GRM5PTGES
SCHEMBL14976213 0.80 FFAR1 (0.42) FFAR1APPADORA2AGRM5ADK
SCHEMBL17714326 0.80 ADK (0.44) MAPTFFAR1APPADORA2AGRM5
SCHEMBL30166211 0.75 SMN1; SMN2 (0.40) MAPTFFAR1PIN1
SCHEMBL24053480 0.75 SMN1; SMN2 (0.37) MAPT
SCHEMBL25274502 0.75 SMN1; SMN2 (0.40) MAPTFFAR1PIN1
SCHEMBL20576176 0.75 APP (0.41) MAPTAPPADORA2AGRM5ADK
SCHEMBL13516538 0.74 GRM5 (0.61) MAPTFFAR1APPADORA2AGRM5
SCHEMBL3441623 0.73 IKBKB (0.45) MAPTGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4153577-A1 NEW MALONITRILE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2023-03-29 EP disclosed
CN-115551837-A Novel malononitrile derivatives 豪夫迈·罗氏有限公司 2022-12-30 CN disclosed