SCHEMBL30107973

SCHEMBL30107973

COc1ccc2c(c1)nnn2-c1cc(-c2ccco2)nc(Cl)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.46
ALDH1A1 P00352 5/20 0.46
HPGD P15428 3/20 0.46
MAPT P10636 3/20 0.46
POLB P06746 3/20 0.46
RAB9A P51151 2/20 0.46
HTT P42858 2/20 0.46
MEN1 O00255 1/20 0.46
THRB P10828 1/20 0.46
ALOX12 P18054 1/20 0.46
PTPN7 P35236 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
KMT2A Q03164 1/20 0.46
MCL1 Q07820 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TSHR P16473 2/20 0.42
HSD17B10 Q99714 2/20 0.42
GAA P10253 1/20 0.42
PTGS1 P23219 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30107951 0.88 PTGS1 (0.46) KDM4EALDH1A1HPGDMAPTPOLB
SCHEMBL30107975 0.80 L3MBTL1 (0.40) KDM4EALDH1A1POLBRAB9AHTT
SCHEMBL30107965 0.76 MET (0.40) KDM4EALDH1A1MAPTPOLBRAB9A
SCHEMBL30108028 0.76 KDM4E (0.43) KDM4EALDH1A1HPGDMCL1TSHR
SCHEMBL30108036 0.75 PIM1 (0.46) KDM4EALDH1A1HPGDMAPTPOLB
SCHEMBL30108039 0.73 ALDH1A1 (0.40) KDM4EALDH1A1HPGDMAPTPOLB
SCHEMBL30107968 0.72 IDH1 (0.35) ALDH1A1POLBRAB9AHTTTDP1
SCHEMBL30107959 0.71 KDM4E (0.44) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL30108012 0.70 TSHR (0.58) KDM4EALDH1A1HPGDPOLBRAB9A
SCHEMBL30107966 0.69 TSHR (0.40) KDM4EALDH1A1MAPTPOLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed