SCHEMBL30108784

SCHEMBL30108784

Cc1cnc(-c2nnc(N[C@@H]3CCCNC3)c3ccccc23)c(O)c1

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.68
CHEK2 O96017 6/20 0.48
IL1B P01584 1/20 0.43
CDK7 P50613 3/20 0.43
CCNH P51946 3/20 0.43
MNAT1 P51948 3/20 0.43
CCNT1 O60563 2/20 0.43
CCNK O75909 2/20 0.43
CDK9 P50750 2/20 0.43
CDK12 Q9NYV4 2/20 0.43
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CHEK1 O14757 6/20 0.42
AURKA O14965 2/20 0.41
RPS6KB1 P23443 2/20 0.41
KCNH2 Q12809 1/20 0.41
PRKCZ Q05513 1/20 0.41
PRKD2 Q9BZL6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28934293 1.00 NLRP3 (0.68) NLRP3CHEK2IL1BCDK7CCNH
SCHEMBL28934289 1.00 NLRP3 (0.68) NLRP3CHEK2IL1BCDK7CCNH
SCHEMBL28934455 0.86 CHEK2 (0.54) NLRP3CHEK2IL1BCDK7CCNH
SCHEMBL30108921 0.86 CHEK2 (0.54) NLRP3CHEK2IL1BCDK7CCNH
SCHEMBL28934459 0.86 CHEK2 (0.54) NLRP3CHEK2IL1BCDK7CCNH
SCHEMBL29131979 0.84 IL1B (0.52) NLRP3CHEK2IL1BCDK7CCNH
SCHEMBL30624974 0.84 IL1B (0.52) NLRP3CHEK2IL1BCDK7CCNH
SCHEMBL29131981 0.84 IL1B (0.52) NLRP3CHEK2IL1BCDK7CCNH
SCHEMBL30108655 0.81 NLRP3 (1.00) NLRP3CHEK2IL1B
SCHEMBL28963200 0.81 NLRP3 (1.00) NLRP3CHEK2IL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed