SCHEMBL30115293

SCHEMBL30115293

FC(F)(F)c1cccnc1-c1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 18/20 0.54
SCN5A Q14524 1/20 0.51
SCN9A Q15858 1/20 0.51
KIF11 P52732 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20983702 0.86 TRPV1 (0.60) TRPV1SCN5ASCN9A
SCHEMBL15624412 0.83 TRPV1 (0.47) TRPV1
SCHEMBL3138189 0.81 CYP2A6 (0.56) TRPV1SCN5ASCN9A
SCHEMBL3702161 0.81 TRPV1 (0.67) TRPV1
SCHEMBL27637538 0.81 TRPV1 (0.52) TRPV1SCN5ASCN9A
SCHEMBL30115268 0.81 CYP2A6 (0.56) TRPV1SCN5ASCN9A
SCHEMBL4972991 0.81 TRPV1 (0.52) TRPV1
SCHEMBL6195448 0.81 TRPV1 (0.56) TRPV1
SCHEMBL9823570 0.79 TRPV1 (0.50) TRPV1
SCHEMBL19072734 0.78 TRPV1 (0.52) TRPV1SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12319683-B2 Azabenzimidazole compounds and pharmaceutical NIPPON SHINYAKU CO., LTD. (JP) 2025-06-03 US disclosed
US-20230002395-A1 AZABENZIMIDAZOLE COMPOUND AND MEDICINE NIPPON SHINYAKU CO., LTD. (JP) 2023-01-05 US disclosed
US-20230000840-A1 THERAPEUTIC AGENTS AND PROPHYLACTIC AGENTS FOR FUNCTIONAL GASTROINTESTINAL DISORDERS AND XEROSTOMIA NIPPON SHINYAKU CO., LTD. (JP) 2023-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230002395-A1 AZABENZIMIDAZOLE COMPOUND AND MEDICINE PAM, CHRM3, AZI2 TRPV1 30/4885SCN5A 1622/4885SCN9A 2513/4885
US-20230000840-A1 THERAPEUTIC AGENTS AND PROPHYLACTIC AGENTS FOR FUNCTIONAL GASTROINTESTINAL DISORDERS AND XEROSTOMIA ALPI, SI, AZI2 TRPV1 624/4885SCN5A 1191/4885SCN9A 2291/4885
US-12319683-B2 Azabenzimidazole compounds and pharmaceutical PAM, CHRM3, AZI2 TRPV1 16/4885SCN5A 835/4885SCN9A 1549/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.