SCHEMBL30122280

SCHEMBL30122280

[2H]C([2H])([2H])n1c(=O)c(Br)cc2c(O)nc(C)nc21

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ESR1 P03372 1/20 0.30
ESRRA P11474 1/20 0.30
ESR2 Q92731 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29861520 0.89 PIK3CA (0.36) PIK3CAKDM4EALDH1A1GLAGAA
SCHEMBL23326861 0.89 PIK3CA (0.36) PIK3CAKDM4EALDH1A1GLAGAA
SCHEMBL30122338 0.80 RXFP1 (0.35) PIK3CAKDM4EALDH1A1GLAGAA
SCHEMBL30122319 0.72 CA1 (0.31)
SCHEMBL23326638 0.71 KDM4E (0.35) PIK3CAKDM4EALDH1A1GLAGAA
SCHEMBL29910267 0.71 KDM4E (0.35) PIK3CAKDM4EALDH1A1GLAGAA
SCHEMBL23326645 0.69 RXFP1 (0.40) PIK3CAKDM4EALDH1A1GLAGAA
SCHEMBL24582788 0.69 CDK4 (0.32)
SCHEMBL29861864 0.69 RXFP1 (0.40) PIK3CAKDM4EALDH1A1GLAGAA
SCHEMBL23326640 0.68 CYP1A2 (0.33) PIK3CAALDH1A1HSD17B10ESR1ESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212531-A1 PYRIDOPYRIMIDINONE COMPOUNDS ACERAND THERAPEUTICS (USA) LIMITED (US) 2022-10-06 WO disclosed