SCHEMBL30129680

SCHEMBL30129680

Cc1ccc2c(-c3ccc(N)c4c3CN(C(=O)OC(C)(C)C)C4=O)cnn2c1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RET P07949 15/20 0.35
ELANE P08246 1/20 0.32
CSNK2A1 P68400 2/20 0.32
CSNK2A2 P19784 1/20 0.32
SCN5A Q14524 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28848982 1.00 RET (0.35) RETELANECSNK2A1CSNK2A2SCN5A
SCHEMBL29879205 0.86 RET (0.38) RETELANECSNK2A1CSNK2A2SCN5A
SCHEMBL28935767 0.78 PIK3CA (0.34) RET
SCHEMBL31484050 0.78 PIK3CA (0.34) RET
SCHEMBL31484164 0.77 MAPT (0.35) RET
SCHEMBL28935785 0.77 MAPT (0.35) RET
SCHEMBL30207696 0.77 MAPT (0.35) RET
SCHEMBL28848960 0.76
SCHEMBL31484108 0.75
SCHEMBL31484084 0.75 MAPT (0.34) RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611925-B HPK1 inhibitors and uses thereof 轩竹生物科技股份有限公司 2025-04-08 CN disclosed
CN-115611925-A HPK1 inhibitors and uses thereof 轩竹生物科技股份有限公司 2023-01-17 CN disclosed
CN-114940683-B HPK1 inhibitors and uses thereof 轩竹(北京)医药科技有限公司 2023-01-17 CN disclosed