SCHEMBL30132771

SCHEMBL30132771

O=C1OC(=Cc2ccncc2)c2ccc(F)cc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
KDM4E B2RXH2 4/20 0.49
TDP1 Q9NUW8 4/20 0.49
HPGD P15428 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
CYP19A1 P11511 2/20 0.47
CYP11B1 P15538 2/20 0.47
CYP11B2 P19099 2/20 0.47
MEN1 O00255 6/20 0.44
KMT2A Q03164 6/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
NFKB1 P19838 1/20 0.44
CYP2C19 P33261 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30132787 0.85 CYP19A1 (0.52) ALDH1A1KDM4ETDP1HPGDL3MBTL1
SCHEMBL7661772 0.81 KDM4E (0.73) ALDH1A1KDM4ETDP1HPGDL3MBTL1
SCHEMBL7661776 0.81 KDM4E (0.73) ALDH1A1KDM4ETDP1HPGDL3MBTL1
SCHEMBL28581666 0.80 KDM4E (0.67) ALDH1A1KDM4ETDP1HPGDL3MBTL1
SCHEMBL2528748 0.77 ALDH1A1 (0.49) ALDH1A1KDM4ETDP1HPGDL3MBTL1
SCHEMBL2528750 0.77 ALDH1A1 (0.49) ALDH1A1KDM4ETDP1HPGDL3MBTL1
SCHEMBL28250731 0.77 KDM4E (0.49) ALDH1A1KDM4ETDP1HPGDL3MBTL1
SCHEMBL28250730 0.77 KDM4E (0.49) ALDH1A1KDM4ETDP1HPGDL3MBTL1
SCHEMBL6586281 0.75 ACHE (0.54) ALDH1A1KDM4ETDP1HPGDCYP19A1
SCHEMBL6586280 0.75 ACHE (0.54) ALDH1A1KDM4ETDP1HPGDCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115485271-A Novel compounds as inhibitors of poly (ADP-ribose) polymerase (PARP) 理森制药股份公司 2022-12-16 CN disclosed