SCHEMBL30135835

SCHEMBL30135835

CCCCOC(=O)NC1CCN(C(=O)CCN2CCN(c3cccc(C4CCC(=O)NC4=O)c3)CC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 5/20 0.41
HTR1A P08908 8/20 0.41
HTR7 P34969 7/20 0.41
DRD2 P14416 1/20 0.39
DDB1 Q16531 4/20 0.39
MAPK1 P28482 1/20 0.39
ADAMTS5 Q9UNA0 1/20 0.38
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
CHRM4 P08173 1/20 0.37
TMEM97 Q5BJF2 2/20 0.37
SIGMAR1 Q99720 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25821980 0.88 DDB1 (0.44) CRBNHTR1AHTR7DRD2DDB1
SCHEMBL30135745 0.88 DDB1 (0.44) CRBNHTR1AHTR7DRD2DDB1
SCHEMBL25031321 0.82 HTR1A (0.49) CRBNHTR1AHTR7DDB1ADAMTS5
SCHEMBL30136072 0.81 TSHR (0.41) CRBNHTR1AHTR7DRD2DDB1
SCHEMBL30135799 0.81 CRBN (0.51) CRBNDRD2DDB1MAPK1CHRM4
SCHEMBL31127674 0.79 CRBN (0.49) CRBNHTR1ADRD2
SCHEMBL25819151 0.79 DDB1 (0.45) CRBNHTR1AHTR7DRD2DDB1
SCHEMBL30822462 0.77 DDB1 (0.51) CRBNHTR1AHTR7DDB1TMEM97
SCHEMBL30135838 0.76 DDB1 (0.51) CRBNHTR1AHTR7DRD2DDB1
SCHEMBL25034990 0.76 DDB1 (0.45) CRBNDRD2DDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4157849-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND Uppthera, Inc. (KR) 2023-04-05 EP disclosed
WO-2023017446-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed
WO-2023018238-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed