SCHEMBL30135865

SCHEMBL30135865

CCCCOC(=O)N1CCC2(CC1)CC(NC(=O)c1cc(OC)c(Nc3ncc4c(n3)N(C(C)C)CC(F)(F)C(=O)N4C)cc1F)C2

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 20/20 0.57
PLK3 Q9H4B4 9/20 0.51
PLK2 Q9NYY3 9/20 0.51
BRD4 O60885 1/20 0.44
BRDT Q58F21 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25334099 0.90 PLK1 (0.63) PLK1PLK3PLK2BRD4BRDT
SCHEMBL25031421 0.89 PLK1 (0.59) PLK1PLK3PLK2BRD4BRDT
SCHEMBL25031422 0.86 PLK1 (0.62) PLK1PLK3PLK2BRD4BRDT
SCHEMBL30135959 0.85 PLK1 (0.54) PLK1PLK3PLK2BRD4BRDT
SCHEMBL30135899 0.83 PLK1 (0.50) PLK1PLK3PLK2BRD4BRDT
SCHEMBL25031487 0.83 PLK1 (0.52) PLK1PLK3PLK2BRD4BRDT
SCHEMBL1675947 0.83 PLK1 (0.80) PLK1PLK3PLK2BRD4BRDT
SCHEMBL30136049 0.83 PLK1 (0.48) PLK1PLK3PLK2BRD4BRDT
SCHEMBL25334301 0.83 PLK1 (0.53) PLK1PLK3PLK2BRD4BRDT
SCHEMBL30135711 0.81 PLK1 (0.71) PLK1PLK3PLK2BRD4BRDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4157850-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND Uppthera, Inc. (KR) 2023-04-05 EP disclosed
WO-2023018236-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed
WO-2023017446-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed