SCHEMBL30135899

SCHEMBL30135899

CCCCOC(=O)N1CCC2(CC1)CC(CNC(=O)c1ccc(Nc3ncc4c(n3)N(C(C)C)CC(F)(F)C(=O)N4C)c(OC)c1)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 20/20 0.50
BRD4 O60885 6/20 0.50
BRDT Q58F21 3/20 0.50
PLK3 Q9H4B4 7/20 0.45
PLK2 Q9NYY3 6/20 0.45
PTK2 Q05397 2/20 0.43
PDXK O00764 1/20 0.43
WEE1 P30291 1/20 0.43
NEK3 P51956 1/20 0.43
CAMKK2 Q96RR4 1/20 0.43
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
PRKCG P05129 1/20 0.42
CLK2 P49760 1/20 0.42
RPS6KA3 P51812 1/20 0.42
NEK4 P51957 1/20 0.42
CAMK2G Q13555 1/20 0.42
CAMK2D Q13557 1/20 0.42
SRPK1 Q96SB4 1/20 0.42
PRKD2 Q9BZL6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30501271 0.90 PLK1 (0.54) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30136049 0.90 PLK1 (0.48) PLK1BRD4BRDTPLK3PLK2
SCHEMBL25935268 0.90 PLK1 (0.52) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30135959 0.87 PLK1 (0.54) PLK1BRD4BRDTPLK3PLK2
SCHEMBL25935265 0.86 PLK1 (0.54) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30136097 0.84 PLK1 (0.67) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30135865 0.83 PLK1 (0.57) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30135947 0.83 PLK1 (0.63) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30135711 0.83 PLK1 (0.71) PLK1BRD4BRDTPLK3PLK2
SCHEMBL25334430 0.81 PLK1 (0.62) PLK1BRD4BRDTPLK3PLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4157850-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND Uppthera, Inc. (KR) 2023-04-05 EP disclosed
WO-2023018236-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed
WO-2023017446-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed