SCHEMBL30136034

SCHEMBL30136034

CCCCOC(=O)NC1CCN(C(=O)CN2CCN(c3ccc(C(=O)NC4CCC(=O)NC4=O)cc3)CC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 8/20 0.44
DDB1 Q16531 3/20 0.44
IKZF3 Q9UKT9 1/20 0.44
KMT2A Q03164 2/20 0.43
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
MAPT P10636 4/20 0.39
ALDH1A1 P00352 1/20 0.39
HIF1A Q16665 1/20 0.39
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
DRD2 P14416 2/20 0.38
PARP1 P09874 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30135938 0.87 CRBN (0.46) CRBNDDB1IKZF3KMT2AHDAC8
SCHEMBL30135743 0.81 CRBN (0.45) CRBNDDB1IKZF3HDAC8DRD2
SCHEMBL29179845 0.80 CRBN (0.49) CRBNDDB1IKZF3KMT2AMAPT
SCHEMBL30135946 0.78 CRBN (0.47) CRBNDDB1IKZF3KMT2ATSHR
SCHEMBL30136072 0.78 TSHR (0.41) CRBNDDB1KMT2AMAPTALDH1A1
SCHEMBL30376308 0.76 CRBN (0.57) CRBNDDB1KMT2AHDAC3HDAC1
SCHEMBL29179871 0.76 CRBN (0.52) CRBNDDB1IKZF3GSPT1
SCHEMBL30135719 0.76 CRBN (0.56) CRBNDDB1IKZF3KMT2AMAPT
SCHEMBL30135835 0.75 CRBN (0.41) CRBNDDB1DRD2
SCHEMBL30965700 0.74 CRBN (0.50) CRBNDDB1KMT2AHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4384521-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND Uppthera, Inc. (KR) 2024-06-19 EP disclosed
WO-2023018237-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed
WO-2023017446-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed