SCHEMBL30137501

SCHEMBL30137501

CC(C)C(=O)Nc1ccc(C(F)(F)F)cc1CN1CCOCC1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.54
L3MBTL1 Q9Y468 2/20 0.51
POLB P06746 1/20 0.51
ALDH1A1 P00352 3/20 0.51
GAA P10253 1/20 0.51
HIF1A Q16665 2/20 0.49
EPAS1 Q99814 2/20 0.49
CNR1 P21554 2/20 0.48
CNR2 P34972 2/20 0.48
LMNA P02545 2/20 0.46
TP53 P04637 1/20 0.46
MGLL Q99685 1/20 0.46
ABHD6 Q9BV23 1/20 0.46
MOK Q9UQ07 1/20 0.46
KDM4E B2RXH2 1/20 0.46
THRB P10828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31053802 0.79 CNR2 (0.45) L3MBTL1POLBALDH1A1HIF1AEPAS1
SCHEMBL25027294 0.79 CNR2 (0.45) L3MBTL1POLBALDH1A1HIF1AEPAS1
SCHEMBL25024820 0.77 CNR2 (0.47) L3MBTL1POLBALDH1A1HIF1AEPAS1
SCHEMBL3445946 0.75 SCN9A (0.52) L3MBTL1POLBALDH1A1HIF1AEPAS1
SCHEMBL30137493 0.74 SMN1; SMN2 (0.48) SMN1; SMN2L3MBTL1ALDH1A1GAALMNA
SCHEMBL24119880 0.73 ALDH1A1 (0.54) SMN1; SMN2ALDH1A1GAALMNATP53
SCHEMBL25026436 0.72 ALOX5AP (0.57) L3MBTL1POLBALDH1A1HIF1AEPAS1
SCHEMBL4242830 0.72 CYP2A13 (0.56) L3MBTL1POLBALDH1A1HIF1AEPAS1
SCHEMBL15915825 0.72 CYP2A13 (0.56) L3MBTL1POLBALDH1A1HIF1AEPAS1
SCHEMBL1977685 0.72 CYP2A13 (0.51) SMN1; SMN2L3MBTL1POLBALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118475567-A Heterocyclic derivative, composition and pharmaceutical application thereof 西藏海思科制药有限公司 2024-08-09 CN disclosed
WO-2023016518-A1 HETEROCYCLIC DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL USE THEREOF 四川海思科制药有限公司 2023-02-16 WO disclosed