SCHEMBL30137586

SCHEMBL30137586

COC(=O)c1ncc(-c2cccc(Cl)c2Cl)nc1NC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.42
PDCD1 Q15116 12/20 0.39
CD274 Q9NZQ7 12/20 0.39
LCK P06239 2/20 0.39
SLC6A3 Q01959 1/20 0.39
PDGFRB P09619 1/20 0.38
FGFR1 P11362 1/20 0.38
SRC P12931 1/20 0.38
PDGFRA P16234 1/20 0.38
ACVR1B P36896 1/20 0.38
TGFBR1 P36897 1/20 0.38
ACVRL1 P37023 1/20 0.38
NUDT1 P36639 1/20 0.38
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31054055 0.91 LCK (0.40) ATRPDCD1CD274LCKPDGFRB
SCHEMBL28967358 0.79 ATR (0.42) ATRLCKSLC6A3PDGFRBFGFR1
SCHEMBL30137565 0.78 NUDT1 (0.44) ATRPDCD1CD274LCKPDGFRB
SCHEMBL22789709 0.77 SLC6A3 (0.44) ATRPDCD1CD274SLC6A3NUDT1
SCHEMBL30683763 0.77 SLC6A3 (0.44) ATRPDCD1CD274SLC6A3NUDT1
SCHEMBL31053916 0.77 LCK (0.43) ATRLCKPDGFRBFGFR1SRC
SCHEMBL20899380 0.75 SLC6A3 (0.43) ATRPDCD1CD274SLC6A3NUDT1
SCHEMBL30137525 0.74 CNR1 (0.41) ATRLCKPDGFRBFGFR1SRC
SCHEMBL28967353 0.74 CNR1 (0.41) ATRLCKPDGFRBFGFR1SRC
SCHEMBL28967339 0.73 CCR4 (0.45) ATRLCKPDGFRBFGFR1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611869-B Heterocyclic pyrazine derivative and application thereof in preparation of SHP2 inhibitor 山东大学 2024-08-09 CN disclosed
CN-115611869-A Heterocyclic pyrazine derivative and application thereof in preparation of SHP2 inhibitor 山东大学 2023-01-17 CN disclosed