SCHEMBL30138283

SCHEMBL30138283

COCCCNc1cc(N)ncn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.46
CYP1A2 P05177 3/20 0.45
CLK4 Q9HAZ1 2/20 0.45
CYP2C19 P33261 2/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
APEX1 P27695 1/20 0.45
CASP7 P55210 1/20 0.45
KDM4E B2RXH2 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX15 P16050 2/20 0.43
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
AURKA O14965 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20929510 1.00 DYRK1A (0.46) DYRK1ACYP1A2CLK4CYP2C19LMNA
SCHEMBL30138398 0.90 CYP1A2 (0.54) CYP1A2CLK4CYP2C19LMNAHTT
SCHEMBL20929509 0.90 CYP1A2 (0.54) CYP1A2CLK4CYP2C19LMNAHTT
SCHEMBL10218021 0.83 CHEK1 (0.50) DYRK1ACYP1A2CLK4CYP2C19LMNA
SCHEMBL18636563 0.81 DNM2 (0.54) CLK4AURKADNM2CHEK1
SCHEMBL17103026 0.80 DNM2 (0.60) CLK4LMNASMN1; SMN2ALDH1A1AURKA
SCHEMBL20929505 0.78 CHEK1 (0.52) DYRK1ACYP1A2CLK4CYP2C19LMNA
SCHEMBL30138380 0.78 CHEK1 (0.52) DYRK1ACYP1A2CLK4CYP2C19LMNA
SCHEMBL10187338 0.78 DNM2 (0.45) HTTALDH1A1AURKADNM2CHEK1
SCHEMBL2231653 0.75 DNM2 (0.48) TSHRAURKADNM2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12472181-B2 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders GALAPAGOS NV (BE) 2025-11-18 US disclosed
US-20230310433-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2023-10-05 US disclosed
US-11564923-B2 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders GALAPAGOS NV (BE) 2023-01-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11564923-B2 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders IL15, IL2, IL33 DYRK1A 3837/4885CYP1A2 275/4885CLK4 2550/4885
US-20230310433-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS IL15, IL2, IL33 DYRK1A 3837/4885CYP1A2 275/4885CLK4 2550/4885
US-12472181-B2 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders IL15, IL2, IL33 DYRK1A 3837/4885CYP1A2 275/4885CLK4 2550/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.