SCHEMBL30139014

SCHEMBL30139014

COC(=O)c1cc(Br)cc2[nH]c(N(Cc3ccccc3)C(=O)OC(C)(C)C)nc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.38
AKT1 P31749 2/20 0.36
MCL1 Q07820 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
PIM1 P11309 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
BACE1 P56817 1/20 0.34
CACNA1G O43497 1/20 0.33
CACNA1B Q00975 1/20 0.33
CACNA1C Q13936 1/20 0.33
STAT5B P51692 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26631541 1.00 DHODH (0.38) DHODHAKT1MCL1KDM4EALDH1A1
SCHEMBL28943154 0.92 DHODH (0.47) DHODHAKT1MCL1STAT5B
SCHEMBL26631532 0.83 CNR1 (0.35) DHODHMCL1KDM4EALDH1A1HPGD
SCHEMBL30138973 0.83 CNR1 (0.35) DHODHMCL1KDM4EALDH1A1HPGD
SCHEMBL23925332 0.75 RNASEH1 (0.50) DHODHKDM4EALDH1A1HPGDCRHBP
SCHEMBL16331805 0.71 AKT1 (0.36) AKT1MCL1HDAC3HDAC1HDAC2
SCHEMBL30138958 0.71 ATR (0.43) DHODHCACNA1BCACNA1C
SCHEMBL20378076 0.71 ATR (0.43) DHODHCACNA1BCACNA1C
SCHEMBL2473065 0.70 TP53 (0.43) AKT1MCL1
SCHEMBL14910299 0.69 KDM4E (0.40) AKT1MCL1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4136077-A1 BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2023-02-22 EP disclosed
CN-115485266-A Benzimidazole derivatives 豪夫迈·罗氏有限公司 2022-12-16 CN disclosed