SCHEMBL30140163

SCHEMBL30140163

Nc1ccc(OC(F)(F)F)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
TSHR P16473 2/20 0.46
SLC1A5 Q15758 2/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
KMO O15229 2/20 0.41
SCN9A Q15858 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
GRIN2B Q13224 2/20 0.39
S100A9 P06702 1/20 0.39
PGK1 P00558 1/20 0.37
ALDH1A1 P00352 1/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
CASP1 P29466 1/20 0.37
RECQL P46063 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL236764 1.00 CYP3A4 (0.46) CYP3A4TSHRSLC1A5CA1CA2
SCHEMBL11298945 0.86 CYP3A4 (0.45) CYP3A4TSHRSLC1A5CA1CA2
SCHEMBL22815715 0.85 KMO (0.47) CYP3A4TSHRSLC1A5KMOGRIN2B
SCHEMBL1555931 0.84 CYP3A4 (0.46) CYP3A4TSHRSLC1A5CA1CA2
SCHEMBL9447561 0.83 MEN1 (0.44) CYP3A4TSHRSLC1A5CA1CA2
SCHEMBL27483990 0.83 CYP3A4 (0.42) CYP3A4TSHRSLC1A5CA1CA2
SCHEMBL3802892 0.82 CYP3A4 (0.48) CYP3A4TSHRCA1CA2MRGPRX4
SCHEMBL9367414 0.81 GAA (0.40) CYP3A4TSHRSCN9AALDH1A1ALOX15
SCHEMBL28351619 0.80 MEN1 (0.42) CYP3A4TSHRSLC1A5CA1CA2
SCHEMBL11307249 0.80 CYP3A4 (0.39) CYP3A4TSHRSLC1A5CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116768824-B Imide azole heterocyclic compound and application thereof 华南农业大学 2025-06-10 CN disclosed
CN-119977850-A Urea derivative containing aryl sulfonamide structure, and preparation method and application thereof 沈阳药科大学 2025-05-13 CN disclosed
CN-112898196-B Potent soluble epoxide hydrolase inhibitors 艾科西斯有限责任公司 2024-12-27 CN disclosed
CN-119060060-A Imidazole-containing ALK2 kinase inhibitors 拜奥克里斯特制药公司 2024-12-03 CN disclosed
CN-110913855-B Imidazole-containing ALK2 kinase inhibitors 拜奥克里斯特制药公司 2024-09-03 CN disclosed
WO-2024129780-A1 BENZIMIDAZOLE DERIVATIVES AS GPX4 INHIBITORS SONATA THERAPEUTICS, INC. (US) 2024-06-20 WO disclosed
CN-112074511-B Substituted benzodiazoles and their use in therapy 托马斯·黑勒戴药物研究基金会 2024-04-26 CN disclosed
CN-111170991-B Antiproliferative compounds and methods of synthesis thereof 细胞基因公司 2023-10-31 CN disclosed
CN-116947740-A Hydroxamic acid compound containing urea structure, preparation method thereof and application of hydroxamic acid compound in preparation of HDAC and sEH dual inhibitors 沈阳药科大学 2023-10-27 CN disclosed
CN-116768824-A Imide azole heterocyclic compound and application thereof 华南农业大学 2023-09-19 CN disclosed
CN-116199636-A 2, 4-disubstituted pyrimidine derivative of targeted tumor immunity kinase, preparation method and application thereof 杭州医学院 2023-06-02 CN disclosed
WO-2022266426-A1 6-(HETEROCYCLOALKYL-OXY)-QUINAZOLINE DERIVATIVES AND USES THEREOF BLACK DIAMOND THERAPEUTICS, INC. (US) 2022-12-22 WO disclosed