SCHEMBL30141430

SCHEMBL30141430

Cc1c(C(C)(F)F)nn(CC2CCC2C(F)(F)F)c1C(=O)Nc1ccnc(C(N)=O)c1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 15/20 0.40
SLC2A1 P11166 1/20 0.37
SLC2A3 P11169 1/20 0.37
SLC2A4 P14672 1/20 0.37
ANO1 Q5XXA6 2/20 0.35
GSK3B P49841 1/20 0.35
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24906235 1.00 SCN10A (0.40) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL24757797 1.00 SCN10A (0.40) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL24906227 1.00 SCN10A (0.40) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL24759025 0.92 SCN10A (0.40) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL24906385 0.92 SCN10A (0.40) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL24906249 0.92 SCN10A (0.40) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL24759024 0.92 SCN10A (0.40) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL24906317 0.88 SCN10A (0.41) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL30141331 0.88 SCN10A (0.41) SCN10ASLC2A1SLC2A3SLC2A4ANO1
SCHEMBL24906515 0.86 SCN10A (0.39) SCN10ASLC2A1SLC2A3SLC2A4ANO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4355733-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2024-04-24 EP claimed
WO-2022263498-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2022-12-22 WO claimed
EP-4355733-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2024-04-24 EP disclosed
WO-2022263498-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2022-12-22 WO disclosed