SCHEMBL30142364

SCHEMBL30142364

CN1CC[C@@H](NC(=O)c2n[nH]c3c(F)cccc23)C1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 16/20 0.57
WNT1 P04628 12/20 0.57
USP30 Q70CQ3 1/20 0.49
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30142335 1.00 DYRK1A (0.57) DYRK1AWNT1USP30NPC1RAB9A
SCHEMBL30142316 0.93 DYRK1A (0.64) DYRK1AWNT1NPC1RAB9A
SCHEMBL30142288 0.82 GSK3B (0.57) DYRK1AWNT1
SCHEMBL30142387 0.82 DYRK1A (0.62) DYRK1AWNT1NPC1RAB9A
SCHEMBL30142298 0.79 GSK3B (0.53) DYRK1AWNT1NPC1RAB9A
SCHEMBL20069732 0.77 L3MBTL1 (0.57) DYRK1AWNT1USP30
SCHEMBL20068957 0.77 KDM5A (0.57) DYRK1AWNT1
SCHEMBL29732688 0.75 NPC1 (0.74) DYRK1AWNT1USP30NPC1RAB9A
SCHEMBL6950689 0.75 NPC1 (0.74) DYRK1AWNT1USP30NPC1RAB9A
SCHEMBL30142314 0.74 GSK3B (0.45) DYRK1AWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220388964-A1 (AZA)INDAZOLYL-ARYL SULFONAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS HIBERCELL, INC. 2022-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220388964-A1 (AZA)INDAZOLYL-ARYL SULFONAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS EIF2AK4, GCN1, GNAI2 DYRK1A 3529/4885WNT1 2112/4885USP30 3469/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.