SCHEMBL30151166

SCHEMBL30151166

Clc1nc(N2CCOCC2)c2oc(CN3CCNCC3)cc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.44
PIK3CB P42338 2/20 0.44
PIK3CD O00329 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SOS1 Q07889 1/20 0.40
PARP1 P09874 1/20 0.39
MTOR P42345 1/20 0.39
PIK3CG P48736 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
PDE7B Q9NP56 1/20 0.38
HRH4 Q9H3N8 5/20 0.36
JAK2 O60674 1/20 0.35
P2RY12 Q9H244 1/20 0.33
CSF1R P07333 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23804721 0.92 SMN1; SMN2 (0.46) PIK3CAPIK3CBPIK3CDSMN1; SMN2PARP1
SCHEMBL4788094 0.87 PIK3CA (0.39) PIK3CAPIK3CBPIK3CDSMN1; SMN2SOS1
SCHEMBL12727282 0.86 PIK3CA (0.46) PIK3CAPIK3CBPIK3CDSMN1; SMN2PARP1
SCHEMBL4752635 0.84 PIK3CA (0.42) PIK3CAPIK3CBPIK3CDSMN1; SMN2PARP1
SCHEMBL2674386 0.82 HRH3 (0.41) PIK3CAPIK3CBPIK3CDSMN1; SMN2PARP1
SCHEMBL189804 0.82 PIK3CA (0.61) PIK3CAPIK3CBPIK3CDMTORPIK3CG
SCHEMBL2673625 0.81 PIK3CD (0.46) PIK3CAPIK3CBPIK3CDPIK3CG
SCHEMBL23804692 0.81 SMN1; SMN2 (0.47) PIK3CAPIK3CBPIK3CDSMN1; SMN2PARP1
SCHEMBL189736 0.80 PIK3CA (0.53) PIK3CAPIK3CBPIK3CDMTORPIK3CG
SCHEMBL12873273 0.79 SMN1; SMN2 (0.43) PIK3CAPIK3CBPIK3CDSMN1; SMN2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113045582-B PARP-1/PI3K double-target inhibitor or pharmaceutically acceptable salt thereof, and preparation method and application thereof 中国药科大学 2022-12-23 CN disclosed