SCHEMBL4788094

SCHEMBL4788094

Clc1nc(N2CCOCC2)c2oc(CN3CC4(CCNCC4)C3)cc2n1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.39
PIK3CB P42338 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
CYP2D6 P10635 4/20 0.38
PIK3CD O00329 2/20 0.37
PDE7B Q9NP56 2/20 0.36
PARP1 P09874 1/20 0.34
MTOR P42345 1/20 0.34
PIK3CG P48736 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
TSHR P16473 1/20 0.34
HRH4 Q9H3N8 4/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
AKT1 P31749 1/20 0.32
SOS1 Q07889 1/20 0.32
HPGD P15428 1/20 0.31
CSF1R P07333 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30151166 0.87 PIK3CA (0.44) PIK3CAPIK3CBSMN1; SMN2PIK3CDPDE7B
SCHEMBL23804721 0.84 SMN1; SMN2 (0.46) PIK3CAPIK3CBSMN1; SMN2PIK3CDPDE7B
SCHEMBL994274 0.82 PIK3CA (0.46) PIK3CAPIK3CBCYP2D6PIK3CDMTOR
SCHEMBL12727282 0.79 PIK3CA (0.46) PIK3CAPIK3CBSMN1; SMN2PIK3CDPARP1
SCHEMBL2674386 0.77 HRH3 (0.41) PIK3CAPIK3CBSMN1; SMN2PIK3CDPDE7B
SCHEMBL13983587 0.77 PIK3CD (0.49) PIK3CAPIK3CBPIK3CDMTORPIK3CG
SCHEMBL12926571 0.77 PIK3CA (0.45) PIK3CAPIK3CBPIK3CDMTORPIK3CG
SCHEMBL4752635 0.76 PIK3CA (0.42) PIK3CAPIK3CBSMN1; SMN2PIK3CDPDE7B
SCHEMBL23804692 0.76 SMN1; SMN2 (0.47) PIK3CAPIK3CBSMN1; SMN2PIK3CDPARP1
SCHEMBL189804 0.75 PIK3CA (0.61) PIK3CAPIK3CBPIK3CDMTORPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008152394-A1 PHARMACEUTICAL COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2008-12-18 WO disclosed