SCHEMBL30158883

SCHEMBL30158883

Cc1ccc(S(=O)(=O)OCCCCCc2ccnc(F)c2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PSMD10 O75832 1/20 0.38
F2 P00734 2/20 0.33
COMT P21964 1/20 0.33
CA12 O43570 4/20 0.33
CA1 P00915 4/20 0.33
CA9 Q16790 4/20 0.33
CA2 P00918 3/20 0.33
GPR119 Q8TDV5 3/20 0.32
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
MMP8 P22894 1/20 0.31
MMP13 P45452 1/20 0.31
STAT3 P40763 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29187914 1.00 PSMD10 (0.38) PSMD10F2COMTCA12CA1
SCHEMBL30158952 0.89 PSMD10 (0.39) PSMD10F2CA12CA1CA9
SCHEMBL29187888 0.89 PSMD10 (0.39) PSMD10F2CA12CA1CA9
SCHEMBL30159151 0.87 PSMD10 (0.37) PSMD10F2CA12CA1CA9
SCHEMBL29187852 0.87 PSMD10 (0.37) PSMD10F2CA12CA1CA9
SCHEMBL28950649 0.84 KMT2A (0.37) PSMD10F2CA12CA1CA9
SCHEMBL28950630 0.84 PSMD10 (0.37) PSMD10CA12CA1CA9CA2
SCHEMBL30159078 0.82 ALDH1A1 (0.43) PSMD10F2COMTCA12CA1
SCHEMBL28950629 0.82 ALDH1A1 (0.43) PSMD10F2COMTCA12CA1
SCHEMBL28950570 0.82 PSMD10 (0.36) PSMD10F2CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-A Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2022-12-30 CN disclosed