SCHEMBL30159062

SCHEMBL30159062

COC(=O)c1cc(OC)n2c(C3CC3)c(-c3ccccn3)nc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
TGFBR1 P36897 2/20 0.38
GRM5 P41594 1/20 0.37
KDM4E B2RXH2 2/20 0.37
MCHR1 Q99705 2/20 0.37
TRPV4 Q9HBA0 1/20 0.36
ALDH1A1 P00352 3/20 0.36
GAA P10253 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALOX15 P16050 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
HTT P42858 2/20 0.36
LMNA P02545 1/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30158931 0.91 JMJD6 (0.36) CYP11B1CYP11B2MCHR1TRPV4MEN1
SCHEMBL30850116 0.84 GRM5 (0.42) TGFBR1GRM5KDM4ETRPV4ALDH1A1
SCHEMBL30159114 0.82 AKT1 (0.46) CYP11B1CYP11B2TGFBR1GRM5KDM4E
SCHEMBL23970744 0.78 ALDH1A1 (0.40) CYP11B1CYP11B2KDM4EALDH1A1SMN1; SMN2
SCHEMBL30850082 0.76 NPC1 (0.48) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL30159083 0.75 KDM4E (0.42) KDM4EALDH1A1GAASMN1; SMN2MEN1
SCHEMBL30159222 0.73 CYP11B1 (0.49) CYP11B1CYP11B2KDM4EMCHR1ALDH1A1
SCHEMBL30158928 0.71 JMJD6 (0.42) CYP11B1CYP11B2TGFBR1MCHR1ALDH1A1
SCHEMBL30850076 0.70 KDM4E (0.38) CYP11B1CYP11B2KDM4EALDH1A1GAA
SCHEMBL15173149 0.69 KDM4E (0.56) TGFBR1GRM5KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-A Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2022-12-30 CN disclosed