SCHEMBL30159083

SCHEMBL30159083

COc1cc(C(=O)O)cc2nc(-c3ccccn3)c(C)n12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
KDM4C Q9H3R0 3/20 0.42
KDM6B O15054 1/20 0.42
KDM4A O75164 1/20 0.42
KDM5C P41229 1/20 0.42
KDM2A Q9Y2K7 1/20 0.42
KDM3A Q9Y4C1 1/20 0.42
KDM5A P29375 2/20 0.40
KDM5B Q9UGL1 1/20 0.40
PIN1 Q13526 1/20 0.40
GAA P10253 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
TP53 P04637 2/20 0.38
NPC1 O15118 2/20 0.38
GABRA5 P31644 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30850116 0.90 GRM5 (0.42) KDM4EKDM4CKDM6BKDM5CKDM2A
SCHEMBL30850082 0.87 NPC1 (0.48) KDM4ESMN1; SMN2NPC1KMT2AMEN1
SCHEMBL30159062 0.75 CYP11B1 (0.39) KDM4EGAASMN1; SMN2TP53NPC1
SCHEMBL30158931 0.72 JMJD6 (0.36) KDM5ANPC1KMT2AMEN1RAB9A
SCHEMBL23971162 0.71 KDM5A (0.38) KDM4EKDM4CKDM5AKDM5BKMT2A
SCHEMBL18311298 0.69 KAT6A (0.64) KDM4EKDM4CKDM6BKDM4AKDM5C
SCHEMBL29642392 0.68 KDM5A (0.43) KDM4CKDM5AKDM5B
SCHEMBL28830424 0.67 KDM4E (0.64) KDM4EKDM4CKDM6BKDM4AKDM5C
SCHEMBL863317 0.67 KDM4E (0.74) KDM4EKDM4CKDM6BKDM4AKDM5C
SCHEMBL28404844 0.67 KDM4E (0.64) KDM4EKDM4CKDM6BKDM4AKDM5C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-B Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2024-04-12 CN disclosed
CN-115551862-A Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2022-12-30 CN disclosed