SCHEMBL30159080

SCHEMBL30159080

C=CC[C@H]1C[C@]1(C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
NR1H3 Q13133 1/20 0.31
PTPN1 P18031 1/20 0.31
APLNR P35414 1/20 0.31
GRM2 Q14416 2/20 0.31
GRM5 P41594 1/20 0.31
GRM1 Q13255 1/20 0.31
RXRA P19793 1/20 0.30
RXRB P28702 1/20 0.30
RXRG P48443 1/20 0.30
FFAR3 O14843 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30159039 1.00 POLB (0.32) POLBMAPTNR1H3PTPN1APLNR
SCHEMBL16826992 0.79 THRB (0.30)
SCHEMBL15483731 0.79 KMT2A (0.32) POLBMAPT
SCHEMBL9397906 0.74 NR1H4 (0.37) POLBMAPTRXRARXRBRXRG
SCHEMBL9397901 0.74 NR1H4 (0.37) POLBMAPTRXRARXRBRXRG
SCHEMBL9397907 0.74 NR1H4 (0.37) POLBMAPTRXRARXRBRXRG
SCHEMBL16506470 0.74
SCHEMBL3152751 0.74
SCHEMBL29188017 0.74
SCHEMBL29188019 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-B Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2024-04-12 CN disclosed
CN-115551862-A Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2022-12-30 CN disclosed