SCHEMBL30161399

SCHEMBL30161399

Cc1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1Br

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.68
CCNB1 P14635 1/20 0.68
CCNA2 P20248 1/20 0.68
CDK2 P24941 1/20 0.68
CDK7 P50613 1/20 0.68
CCNH P51946 1/20 0.68
CCNA1 P78396 1/20 0.68
ALDH1A1 P00352 5/20 0.62
LMNA P02545 2/20 0.62
MAPT P10636 3/20 0.59
HTT P42858 2/20 0.59
MAPK1 P28482 1/20 0.56
HPGD P15428 2/20 0.54
HSD17B10 Q99714 1/20 0.54
MCL1 Q07820 4/20 0.54
EDNRB P24530 2/20 0.53
EDNRA P25101 2/20 0.53
HSP90AA1 P07900 1/20 0.53
HSP90AB1 P08238 1/20 0.53
TP53 P04637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25453798 1.00 CDK1 (0.68) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL13615072 0.80 CDK1 (0.63) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL13629329 0.80 ALDH1A1 (0.65) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL14403379 0.77 MEN1 (0.62) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL16325537 0.75 CDK1 (0.65) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL31689483 0.75 CES1 (0.62) ALDH1A1MAPTTDP1IDH1
SCHEMBL29561662 0.75 PKM (0.53)
SCHEMBL22095989 0.75 MAPK1 (0.71) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL29118839 0.75 ALDH1A1 (0.67) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL95927 0.75 ALDH1A1 (0.67) CDK1CCNB1CCNA2CDK2CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115768750-A GCN2 modulator compounds 阿莱斯塔治疗公司 2023-03-07 CN disclosed
EP-4107146-A1 GCN2 MODULATOR COMPOUNDS Alesta Therapeutics BV (NL) 2022-12-28 EP disclosed