Estradiol Propionate

Estradiol Propionate

SCHEMBL30165166

CCC(=O)O[C@H]1CC[C@H]2[C@@H]3CCc4cc(O)ccc4[C@H]3CC[C@]12C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 1.00
KMT2A Q03164 7/20 1.00
MEN1 O00255 6/20 1.00
CYP3A4 P08684 6/20 1.00
TP53 P04637 4/20 1.00
ALOX15 P16050 3/20 1.00
MAPK1 P28482 3/20 1.00
LMNA P02545 7/20 0.82
ESR1 P03372 5/20 0.82
SMN1; SMN2 Q16637 3/20 0.82
PGR P06401 2/20 0.82
ADORA3 P0DMS8 2/20 0.82
AR P10275 2/20 0.82
PTGS1 P23219 2/20 0.82
PDE3A Q14432 2/20 0.82
POLB P06746 1/20 0.82
CHRM1 P11229 1/20 0.82
TBXA2R P21731 1/20 0.82
ATM Q13315 1/20 0.82
USP2 O75604 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Estradiol Propionate SCHEMBL26659949 1.00 MAPT (1.00) MAPTKMT2AMEN1CYP3A4TP53
Estradiol Propionate SCHEMBL480992 1.00 MAPT (1.00) MAPTKMT2AMEN1CYP3A4TP53
Estradiol Propionate SCHEMBL30384276 1.00 MAPT (1.00) MAPTKMT2AMEN1CYP3A4TP53
Estradiol Propionate SCHEMBL28094685 0.98 MAPT (0.96) MAPTKMT2AMEN1CYP3A4TP53
Estradiol Propionate SCHEMBL28092621 0.95 MAPT (0.91) MAPTKMT2AMEN1CYP3A4TP53
Estradiol Propionate SCHEMBL27583398 0.93 MAPT (0.86) MAPTKMT2AMEN1CYP3A4TP53
SCHEMBL9404746 0.92 MAPT (0.89) MAPTKMT2AMEN1CYP3A4TP53
SCHEMBL19393249 0.92 MAPT (0.89) MAPTKMT2AMEN1CYP3A4TP53
SCHEMBL822184 0.92 MAPT (0.85) MAPTKMT2AMEN1CYP3A4TP53
SCHEMBL19286812 0.92 MAPT (0.85) MAPTKMT2AMEN1CYP3A4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4688003-A2 LIPOSOMAL COMPOSITIONS OF ARCHEXIN The Whiteoak Group, Inc. (US) 2026-02-11 EP disclosed
EP-4630562-A1 NUCLEIC ACID BASED CANCER VACCINE AND METHODS THEREOF Advanced RNA Vaccine (ARV) Technologies, Inc. (US) 2025-10-15 EP disclosed
EP-4608812-A1 VITAMIN-BASED LIPIDS AND LIPID NANOPARTICLES COMPRISING THE SAME Advanced RNA Vaccine (ARV) Technologies, Inc. (US) 2025-09-03 EP disclosed
EP-4577193-A1 COMPOSITIONS AND METHODS FOR THE DELIVERY OF ACTIVE AGENTS INCLUDING NUCLEIC ACIDS Ohio State Innovation Foundation (US) 2025-07-02 EP disclosed
EP-4568645-A2 STEROL BASED IONIZABLE LIPIDS AND LIPID NANOPARTICLES COMPRISING THE SAME Advanced RNA Vaccine (ARV) Technologies, Inc. (US) 2025-06-18 EP disclosed
WO-2024206077-A2 DOSING REGIMES AND COMBINATION THERAPIES USING ARCHEXIN FOR THE TREATMENT OF CANCER THE WHITEOAK GROUP, INC. (US) 2024-10-03 WO disclosed
WO-2024206078-A2 LIPOSOMAL COMPOSITIONS OF ARCHEXIN THE WHITEOAK GROUP, INC. (US) 2024-10-03 WO disclosed
WO-2024124232-A1 NUCLEIC ACID BASED CANCER VACCINE AND METHODS THEREOF ADVANCED RNA VACCINE (ARV) TECHNOLOGIES, INC. (US) 2024-06-13 WO disclosed
WO-2024092209-A1 VITAMIN-BASED LIPIDS AND LIPID NANOPARTICLES COMPRISING THE SAME ADVANCED RNA VACCINE (ARV) TECHNOLOGIES, INC. (US) 2024-05-02 WO disclosed
WO-2024044370-A1 COMPOSITIONS AND METHODS FOR THE DELIVERY OF ACTIVE AGENTS INCLUDING NUCLEIC ACIDS OHIO STATE INNOVATION FOUNDATION (US) 2024-02-29 WO disclosed
WO-2024035710-A2 STEROL BASED IONIZABLE LIPIDS AND LIPID NANOPARTICLES COMPRISING THE SAME ADVANCED RNA VACCINE (ARV) TECHNOLOGIES, INC. (US) 2024-02-15 WO disclosed
WO-2023133560-A2 TISSUE ENGINEERING AND DRUG DELIVERY DEVICE OHIO STATE INNOVATION FOUNDATION (US) 2023-07-13 WO disclosed
WO-2022271255-A1 TISSUE-ENGINEERED SCAFFOLDS AND METHODS OF MAKING GEORGIA TECH RESEARCH CORPORATION (US) 2022-12-29 WO disclosed