SCHEMBL30171244

SCHEMBL30171244

Cn1c(=O)n(CCCO)c(=O)c2c1nc(-c1cccc(OC(F)(F)F)c1)n2Cc1ccc(Cl)cn1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPC5 Q9UL62 16/20 0.63
TRPC4 Q9UBN4 2/20 0.63
TRPC1 P48995 1/20 0.63
KCNH2 Q12809 1/20 0.51
PCSK9 Q8NBP7 1/20 0.45
ADORA2A P29274 2/20 0.44
GRIN1 Q05586 1/20 0.42
GRIN2B Q13224 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16076259 1.00 TRPC5 (0.63) TRPC5TRPC4TRPC1KCNH2PCSK9
SCHEMBL30171322 0.91 TRPC5 (0.56) TRPC5TRPC4TRPC1KCNH2PCSK9
SCHEMBL16076067 0.91 TRPC5 (0.56) TRPC5TRPC4TRPC1KCNH2PCSK9
SCHEMBL16028531 0.90 TRPC5 (0.77) TRPC5TRPC4TRPC1KCNH2PCSK9
SCHEMBL30171267 0.88 TRPC5 (0.49) TRPC5TRPC4TRPC1KCNH2GRIN1
SCHEMBL16076068 0.88 TRPC5 (0.49) TRPC5TRPC4TRPC1KCNH2GRIN1
SCHEMBL30171205 0.88 TRPC5 (0.51) TRPC5TRPC4TRPC1KCNH2GRIN1
SCHEMBL16076095 0.88 TRPC5 (0.56) TRPC5TRPC4TRPC1KCNH2GRIN1
SCHEMBL30171356 0.88 TRPC5 (0.56) TRPC5TRPC4TRPC1KCNH2GRIN1
SCHEMBL16028070 0.88 TRPC5 (0.51) TRPC5TRPC4TRPC1KCNH2GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250034143-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES, LLC (US) 2025-01-30 US disclosed
US-11958854-B2 Substituted xanthines and methods of use thereof HYDRA BIOSCIENCES, LLC (US) 2024-04-16 US disclosed
US-20230040259-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES, LLC (US) 2023-02-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11958854-B2 Substituted xanthines and methods of use thereof TRPC5, TRPC7, TRPC4 TRPC5 1/4885TRPC4 3/4885TRPC1 4/4885
US-20230040259-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF TRPC5, TRPC7, TRPC4 TRPC5 1/4885TRPC4 3/4885TRPC1 4/4885
US-20250034143-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF TRPC5, TRPC7, TRPC4 TRPC5 1/4885TRPC4 3/4885TRPC1 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.