SCHEMBL30176308

SCHEMBL30176308

N#Cc1c(C2CCOCC2)n(-c2ccc(F)cc2)c2ccc(OCc3ccccc3)cc12

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AS3MT Q9HBK9 3/20 0.47
SCN9A Q15858 1/20 0.41
CNR1 P21554 2/20 0.40
CNR2 P34972 2/20 0.40
NSD2 O96028 1/20 0.40
EDNRB P24530 2/20 0.39
EDNRA P25101 2/20 0.39
MAOB P27338 3/20 0.38
MAOA P21397 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RORC P51449 2/20 0.38
PRKDC P78527 1/20 0.35
MCHR1 Q99705 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23886826 1.00 AS3MT (0.47) AS3MTSCN9ACNR1CNR2NSD2
SCHEMBL28995442 0.82 SCN9A (0.40) SCN9ACNR1CNR2ALDH1A1TSHR
SCHEMBL30176384 0.81 SCN9A (0.36) SCN9ACNR1CNR2ALDH1A1TSHR
SCHEMBL23887039 0.81 SCN9A (0.36) SCN9ACNR1CNR2ALDH1A1TSHR
SCHEMBL23886968 0.80 AS3MT (0.54) AS3MTNSD2EDNRBEDNRAMAOB
SCHEMBL30337805 0.79 SCN9A (0.45) SCN9ACNR1CNR2ALDH1A1RORC
SCHEMBL23886885 0.78 SCN9A (0.47) SCN9ACNR1CNR2MAOBMAOA
SCHEMBL30337752 0.78 SCN9A (0.47) SCN9ACNR1CNR2MAOBMAOA
SCHEMBL23898529 0.77 GAA (0.42) CNR1CNR2ALDH1A1TSHRL3MBTL1
SCHEMBL23898492 0.76 CNR1 (0.41) AS3MTCNR1CNR2EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916749-A Substituted 5-hydroxyindole compounds as alpha-1 antitrypsin modulators 弗特克斯药品有限公司 2023-04-04 CN disclosed
EP-4126817-A1 SUBSTITUTED 5-HYDROXYINDOLE COMPOUNDS AS MODULATORS OF ALPHA-1 ANTITRYPSIN Vertex Pharmaceuticals Incorporated (US) 2023-02-08 EP disclosed