SCHEMBL30183161

SCHEMBL30183161

CC1(C)Cc2cnc(N)nc2-c2[nH]nc(C(=O)Nc3nc(C4(C(=O)O)CC4)cs3)c21

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 4/20 0.40
PDE1A P54750 2/20 0.34
PDE1B Q01064 2/20 0.34
PDE1C Q14123 2/20 0.34
CDK4 P11802 1/20 0.30
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CCND3 P30281 1/20 0.30
CDK6 Q00534 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20649344 1.00 PDE5A (0.40) PDE5APDE1APDE1BPDE1CCDK4
SCHEMBL20648980 0.92 PDE5A (0.34) PDE5APDE1APDE1BPDE1C
SCHEMBL30183286 0.86 L3MBTL1 (0.38) CDK4CCNA2CDK2CCND3CDK6
SCHEMBL20649193 0.86 L3MBTL1 (0.38) CDK4CCNA2CDK2CCND3CDK6
SCHEMBL20648932 0.86 GRM5 (0.40)
SCHEMBL30183122 0.86 GRM5 (0.40)
SCHEMBL30183295 0.84 CSNK2A1 (0.40) PDE5A
SCHEMBL20649369 0.84 CSNK2A1 (0.40) PDE5A
SCHEMBL20649045 0.84 CSNK2A1 (0.37) PDE5ACDK2
SCHEMBL30183497 0.84 ATR (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997678-B Pyrazoloquinazoline derivatives as choline kinase inhibitors 内尔维亚诺医疗科学公司 2023-02-21 CN claimed
CN-110997678-B Pyrazoloquinazoline derivatives as choline kinase inhibitors 内尔维亚诺医疗科学公司 2023-02-21 CN disclosed