SCHEMBL30185550

SCHEMBL30185550

Cc1nc(N=C(c2ccccc2)c2ccccc2)sc1-c1ccc2c(c1)C(C(F)(F)F)=NC2=O

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 6/20 0.32
HRH2 P25021 3/20 0.31
HRH1 P35367 3/20 0.31
HRH4 Q9H3N8 3/20 0.31
HRH3 Q9Y5N1 3/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PIK3CD O00329 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
PIK3CG P48736 1/20 0.31
PI4KB Q9UBF8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29099605 1.00 GPR52 (0.32) GPR52HRH2HRH1HRH4HRH3
SCHEMBL30185551 0.82 TSHR (0.32) GPR52NPC1ALDH1A1MAPTHPGD
SCHEMBL30185591 0.77 HRH2 (0.36) GPR52HRH2HRH1HRH4HRH3
SCHEMBL29099535 0.77 HRH2 (0.36) GPR52HRH2HRH1HRH4HRH3
SCHEMBL3085308 0.72 PIK3CD (0.52) NPC1ALDH1A1MAPTHPGDRAB9A
SCHEMBL24023265 0.71 PIK3CA (0.31) HRH2HRH1HRH4HRH3PIK3CA
SCHEMBL24023393 0.71 PIK3CA (0.48) PIK3CDPIK3CAPIK3CBPIK3CGPI4KB
SCHEMBL24023268 0.70 MEN1 (0.33) NPC1ALDH1A1MAPTHPGDRAB9A
SCHEMBL24023338 0.68 XIAP (0.34) NPC1ALDH1A1HPGDRAB9A
SCHEMBL24023335 0.68 PIK3CA (0.41) ALDH1A1MAPTRAB9ASMN1; SMN2PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611883-B PI3K alpha inhibitor with double-ring structure, and preparation method and application thereof 生物岛实验室 2025-03-28 CN disclosed
CN-115611883-A PI3K alpha inhibitor with bicyclic structure and preparation method and application thereof 生物岛实验室 2023-01-17 CN disclosed