SCHEMBL30185551

SCHEMBL30185551

Cc1nc(N=C(c2ccccc2)c2ccccc2)sc1-c1cccc2c1C(C(F)(F)F)=NC2=O

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.32
GPR52 Q9Y2T5 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29099605 0.82 GPR52 (0.32) GPR52NPC1ALDH1A1MAPTHPGD
SCHEMBL30185550 0.82 GPR52 (0.32) GPR52NPC1ALDH1A1MAPTHPGD
SCHEMBL30185559 0.77 MPL (0.39) GPR52NPC1ALDH1A1MAPTHPGD
SCHEMBL24023265 0.67 PIK3CA (0.31)
SCHEMBL3085308 0.66 PIK3CD (0.52) NPC1ALDH1A1MAPTHPGDRAB9A
SCHEMBL24023268 0.65 MEN1 (0.33) TSHRNPC1ALDH1A1MAPTHPGD
SCHEMBL14302479 0.64 SMN1; SMN2 (0.36) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL24023331 0.64 ALDH1A1 (0.36) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL3086729 0.64 ALDH1A1 (0.36) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL24023393 0.64 PIK3CA (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611883-A PI3K alpha inhibitor with bicyclic structure and preparation method and application thereof 生物岛实验室 2023-01-17 CN disclosed