SCHEMBL30185564

SCHEMBL30185564

CCOC(=O)C=C(c1cccc(Br)c1)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 3/20 0.42
MAPK1 P28482 1/20 0.42
LMNA P02545 2/20 0.41
TSHR P16473 1/20 0.41
ELANE P08246 3/20 0.41
RXFP1 Q9HBX9 1/20 0.41
PARP1 P09874 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 2/20 0.40
CYP19A1 P11511 1/20 0.40
HPGD P15428 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30185573 1.00 ALDH1A1 (0.46) ALDH1A1MAPTKDM4EMAPK1LMNA
SCHEMBL30935225 1.00 ALDH1A1 (0.46) ALDH1A1MAPTKDM4EMAPK1LMNA
SCHEMBL29099596 1.00 ALDH1A1 (0.46) ALDH1A1MAPTKDM4EMAPK1LMNA
SCHEMBL29099498 1.00 ALDH1A1 (0.46) ALDH1A1MAPTKDM4EMAPK1LMNA
SCHEMBL29867506 0.86 NPC1 (0.48) ALDH1A1MAPTKDM4EMAPK1LMNA
SCHEMBL23124816 0.85 NQO2 (0.49) ALDH1A1MAPTRAB9AGAAPOLB
SCHEMBL15280988 0.85 CES2 (0.49) ALDH1A1MAPTKDM4ELMNATSHR
SCHEMBL23124814 0.85 NQO2 (0.49) ALDH1A1MAPTRAB9AGAAPOLB
SCHEMBL1274890 0.84 MAPT (0.47) ALDH1A1MAPTMAPK1LMNATSHR
SCHEMBL1274891 0.84 MAPT (0.47) ALDH1A1MAPTMAPK1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611883-A PI3K alpha inhibitor with bicyclic structure and preparation method and application thereof 生物岛实验室 2023-01-17 CN disclosed