SCHEMBL30185655

SCHEMBL30185655

COC(=O)Nc1cc(-c2cc(C(F)F)c(F)cn2)ccn1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 18/20 0.64
CYP3A4 P08684 3/20 0.51
GAK O14976 2/20 0.51
ROCK2 O75116 2/20 0.51
CIT O14578 1/20 0.51
MKNK1 Q9BUB5 1/20 0.51
MYLK2 Q9H1R3 1/20 0.51
TNIK Q9UKE5 1/20 0.51
PIK3C3 Q8NEB9 2/20 0.49
DAPK3 O43293 1/20 0.48
JAK2 O60674 1/20 0.48
DAPK1 P53355 1/20 0.48
TYRO3 Q06418 1/20 0.48
DMPK Q09013 1/20 0.48
HIPK4 Q8NE63 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48
BMP2K Q9NSY1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29174170 0.81 AAK1 (0.61) AAK1CYP3A4GAKROCK2PIK3C3
SCHEMBL30185615 0.81 AAK1 (0.61) AAK1CYP3A4GAKROCK2PIK3C3
SCHEMBL24897652 0.80 AAK1 (0.62) AAK1CYP3A4GAKROCK2CIT
SCHEMBL30185619 0.80 AAK1 (0.62) AAK1CYP3A4GAKROCK2CIT
SCHEMBL17155570 0.79 AAK1 (1.00) AAK1CYP3A4GAKROCK2CIT
SCHEMBL20738221 0.79 AAK1 (1.00) AAK1CYP3A4GAKROCK2CIT
SCHEMBL29400561 0.79 AAK1 (1.00) AAK1CYP3A4GAKROCK2CIT
SCHEMBL30059554 0.78 AAK1 (1.00) AAK1CYP3A4GAKROCK2CIT
SCHEMBL20154451 0.78 AAK1 (1.00) AAK1CYP3A4GAKROCK2CIT
SCHEMBL30185610 0.78 AAK1 (0.81) AAK1CYP3A4GAKROCK2CIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023284838-A1 AAK1 INHIBITOR AND USE THEREOF 四川海思科制药有限公司 2023-01-19 WO disclosed