SCHEMBL24897652

SCHEMBL24897652

COC(=O)Nc1cc(-c2ccc(F)c(C(F)F)n2)ccn1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 18/20 0.62
DAPK1 P53355 3/20 0.62
MKNK2 Q9HBH9 3/20 0.62
BMP2K Q9NSY1 3/20 0.62
GAK O14976 2/20 0.62
DAPK3 O43293 2/20 0.62
JAK2 O60674 2/20 0.62
HIPK4 Q8NE63 2/20 0.62
ROCK2 O75116 1/20 0.62
TYRO3 Q06418 1/20 0.62
DMPK Q09013 1/20 0.62
MKNK1 Q9BUB5 2/20 0.50
MYLK2 Q9H1R3 2/20 0.50
CIT O14578 1/20 0.50
MAP2K1 Q02750 1/20 0.50
PKN2 Q16513 1/20 0.50
TLK2 Q86UE8 1/20 0.50
STK39 Q9UEW8 1/20 0.50
TLK1 Q9UKI8 1/20 0.50
HTR2B P41595 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30185619 1.00 AAK1 (0.62) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL30185629 0.89 TGFBR1 (0.56) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL24897650 0.89 TGFBR1 (0.56) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL27220598 0.87 AAK1 (0.48) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL24897751 0.84 AAK1 (0.58) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL30921024 0.84 AAK1 (0.58) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL30185655 0.80 AAK1 (0.64) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL20447192 0.80 AAK1 (0.61) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL24897623 0.78 AAK1 (0.78) AAK1DAPK1MKNK2BMP2KGAK
SCHEMBL24897655 0.78 AAK1 (0.78) AAK1DAPK1MKNK2BMP2KGAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117715899-A AAK1 inhibitors and uses thereof 西藏海思科制药有限公司 2024-03-15 CN disclosed
WO-2023284838-A1 AAK1 INHIBITOR AND USE THEREOF 四川海思科制药有限公司 2023-01-19 WO disclosed