SCHEMBL30187789

SCHEMBL30187789

COC(C)c1ccc(C#N)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.46
CYP2A6 P11509 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.40
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
TSHR P16473 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11032485 0.94 KIF11 (0.46) CYP19A1CYP2A6ALDH1A1CA12CA2
SCHEMBL1338710 0.81 AKR1C2 (0.42) ALDH1A1CYP11B1CYP11B2TSHRL3MBTL1
SCHEMBL7385564 0.80 CYP2A6 (0.46) CYP19A1CYP2A6ALDH1A1HTTCA12
SCHEMBL2266164 0.80 CYP2A6 (0.46) CYP19A1CYP2A6ALDH1A1HTTCA12
SCHEMBL27480613 0.79 CYP2A6 (0.41) CYP19A1CYP2A6ALDH1A1HTTCA12
SCHEMBL19122181 0.78 HDAC8 (0.37) CA12CA2CA9CA14HDAC8
SCHEMBL5538506 0.78 CYP2A6 (0.40) CYP19A1CYP2A6ALDH1A1HTTCA12
SCHEMBL22824023 0.78 CYP2A6 (0.45) CYP19A1CYP2A6ALDH1A1HTTCA12
SCHEMBL6077332 0.77 CYP2A6 (0.43) CYP19A1CYP2A6ALDH1A1HTTCA12
SCHEMBL6205272 0.77 CYP2A6 (0.43) CYP19A1CYP2A6ALDH1A1HTTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109310668-B Positive allosteric modulators of muscarinic acetylcholine receptor M4 范德比尔特大学 2023-01-24 CN disclosed